Theme


NSAID gastroprotection · Phase III clinical evidence

Tegoprazan vs lansoprazole for preventing NSAID-related peptic ulcers

Source
Source: Gut Liver online-ahead-of-print phase III randomized, double-blind, active-controlled, multicenter study of tegoprazan for prevention of NSAID-induced peptic ulcer in patients on long-term NSAID therapy. The publication cites ClinicalTrials.gov identifier NCT04840550.

Tegoprazan matched lansoprazole for preventing NSAID-related peptic ulcers over 24 weeks, with comparable safety.

Study at a glance

Active-controlled, physician-relevant comparator
Design
Randomized, double-blind, multicenter Phase III
Population
Long-term NSAID users requiring ulcer prevention
Arms
Tegoprazan 25 mg vs lansoprazole 15 mg
Follow-up
Up to 24 weeks
Primary efficacy endpoint
Week 24 peptic ulcer incidence
Non-inferior
Tegoprazan 25 mg met the non-inferiority criterion versus lansoprazole 15 mg for prevention of NSAID-induced gastroduodenal ulcers.
p=0.0004
Primary endpoint met
24
Weeks of ulcer prevention follow-up
Why prevention matters

Chronic NSAID exposure raises gastroduodenal ulcer risk

Long-term NSAID therapy can compromise upper gastrointestinal mucosal protection. For patients who need continuous NSAIDs, proactive acid suppression is a key strategy to reduce peptic ulcer development.

Clinical context
Continuous NSAID users often require durable gastroprotection.
Clinical question
Can tegoprazan provide ulcer prevention comparable to lansoprazole?

Key findings by endpoint

Per-protocol efficacy analysis: 269 patients
Endpoint Timing Finding Reported statistic
Peptic ulcer incidence Week 24 Tegoprazan non-inferior to lansoprazole p=0.0004
Heartburn-free rate Week 12 Favored tegoprazan Direction reported; rate not specified in provided data
Adverse drug reactions Up to 24 weeks Comparable between groups No significant difference reported
Serious adverse events Up to 24 weeks Comparable between groups No significant difference reported
392
Patients randomized 1:1
269
Included in per-protocol analysis
25 mg vs 15 mg
Tegoprazan dose compared with lansoprazole
Clinical takeaway

For patients requiring continuous long-term NSAID therapy, tegoprazan 25 mg appears to be a clinically effective and well-tolerated alternative to lansoprazole 15 mg for peptic ulcer prevention.

AbbreviationsQuick
Abbreviations: ADRs, adverse drug reactions; NSAIDs, nonsteroidal anti-inflammatory drugs; SAEs, serious adverse events.
Bibliography1
  1. Kim SG, Kim TO, Jung SW, et al. A Phase III, Randomized, Double-Blind, Active-Controlled, Multicenter Study Evaluating the Safety and Efficacy of Tegoprazan for the Prevention of Peptic Ulcer in Patients on Continuous Long-Term Treatment with Nonsteroidal Anti-Inflammatory Drugs. Gut Liver. Published online June 22, 2026. doi:10.5009/gnl260057 (DOI: 10.5009/gnl260057)